IB Chemistry R3.4 R3.4.9

Mechanisms of Nucleophilic Substitution

Full SN1 and SN2 mechanisms with stereochemistry: Walden inversion and racemic mixtures.

Reactivity 3.4 HL Extension ⏱️ ~5 min revision
HL Extension

SN1 vs SN2 Mechanistic Overview

Nucleophilic substitution proceeds via two distinct mechanistic pathways depending on the steric and electronic structure of the halogenoalkane substrate:

  • \(\text{S}_\text{N}2\): Bimolecular, concerted 1-step mechanism (favoured by 1° halogenoalkanes).
  • \(\text{S}_\text{N}1\): Unimolecular, 2-step mechanism via carbocation intermediate (favoured by 3° halogenoalkanes).

The SN2 Mechanism

SN2: Concerted Backside Attack

R3.4.9 Mechanisms of Nucleophilic Substitution | ChemEasy HO⁻ C Br H H CH₃ Backside attack C HO δ− Br δ− H H CH₃ Planar TS HO C H CH₃ H + Br⁻ Inverted
SN2 Pathway

SN2 Mechanism: Concerted Backside Attack

  1. Nucleophile attacks \(\text{C}^{\delta+}\) from the opposite side of the leaving group (backside attack, 180°).
  2. Passes through an unstable five-coordinate transition state \([\text{Nu}\cdots\text{C}\cdots\text{X}]^\ddagger\) with negative charge delocalised.
  3. Causes complete inversion of configuration (Walden inversion, like an umbrella turning inside out).

The SN1 Mechanism

SN1 Pathway

SN1 Mechanism: Two-Step Carbocation Pathway

  1. Step 1 (Slow, RDS): Heterolytic fission of \(\text{C}-\text{X}\) bond → planar carbocation intermediate formed.
  2. Step 2 (Fast): Nucleophile attacks planar \(\text{C}^+\) with equal 50% probability from either face → racemic mixture (loss of optical activity).

SN1 vs SN2 Comparison

SN1 SN2
Steps2 (carbocation intermediate)1 (concerted)
SubstrateTertiary halogenoalkanesPrimary halogenoalkanes
StereochemistryRacemic mixtureInversion (Walden)
NucleophileWeak (e.g. H₂O)Strong (e.g. OH⁻)
Secondary substratesBoth mechanisms can occur

Why Does Substrate Type Matter?

HL Extension

Substrate Preference Explanation

Tertiary (3°) → SN1

Bulky alkyl groups cause steric hindrance preventing backside attack, but stabilise the \(3^\circ\) carbocation intermediate via \(+I\) inductive effect.

Primary (1°) → SN2

Minimal steric hindrance allows easy backside attack; a \(1^\circ\) carbocation is too unstable to form via \(\text{S}_\text{N}1\).

Key Insight

Molecularity in Reaction Nomenclature

The numbers "1" and "2" in \(\text{S}_\text{N}1\) and \(\text{S}_\text{N}2\) refer to molecularity (the number of reactant particles in the rate-determining step), NOT the number of steps in the reaction!

Examiner Trap

Stereochemical and Mechanism Pitfalls

  • Transition state brackets: For \(\text{S}_\text{N}2\), always draw square brackets with dotted partial bonds and a negative superscript \([\cdots]^-\).
  • Stereochemistry: \(\text{S}_\text{N}2\) yields inversion; \(\text{S}_\text{N}1\) yields a racemic mixture.
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