IB Chemistry R3.4 R3.4.9
R3.4.9 HL

Electrophilic Substitution

Nitration and halogenation of benzene using Lewis acid catalysts.

📘 IB Understanding

Benzene undergoes electrophilic substitution rather than addition. This preserves the thermodynamic stability of the delocalised π-system. A Lewis acid catalyst generates the electrophile.

Nitration of Benzene

Conditions

Concentrated HNO₃ + concentrated H₂SO₄ at 50 °C

Electrophile Generation

HNO₃ + H₂SO₄ → NO₂⁺ + HSO₄⁻ + H₂O

The nitronium ion (NO₂⁺) is the electrophile.

Halogenation of Benzene

Conditions

Cl₂ or Br₂ with a Lewis acid catalyst (AlCl₃, AlBr₃, or FeBr₃)

Electrophile Generation

Br₂ + AlBr₃ → Br⁺ + AlBr₄⁻

The Lewis acid polarises the halogen molecule, generating the Br⁺ electrophile.

The General Mechanism

  1. The electrophile (E⁺) attacks the delocalised π-system of benzene
  2. A C–E bond forms, creating a positively charged intermediate (arenium ion)
  3. A proton (H⁺) is lost, restoring the aromatic ring

📋 Exam Tip

Always show the curly arrow from the benzene ring (π-electrons) to the electrophile in step 1. The ring acts as the nucleophile. Show the loss of H⁺ in the final step to restore aromaticity.

← R3.4.8 Electrophilic AdditionR3.4.10 Elimination Reactions →